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(+)-UH 232 maleate Please inquire  | Purity Not Available

BOC Sciences

(+)-UH 232 maleate is a dopamine D2 antagonist (Ki = 72.7 nM in a ligand binding assay; apparent KB = 14.5 nM in a cAMP accumulation assay) that preferentially effects on central dopamine autoreceptors. (+)-UH 232 maleate significantly promotes dopamine synthesis and turnover. (+)-UH 232 maleate is also a dopamine D3 partial agonist.

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