Palomid 529 (P529) 50mg | Purity Not Available
Selleck Chemicals
Palomid 529 (P529, SG 00529) inhibits both the mTORC1 and mTORC2 complexes, reduces phosphorylation of pAktS473, pGSK3βS9, and pS6. Phase 1.
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UK 383367 10mg | Purity Not Available
Selleck Chemicals
UK-383367 is a procollagen C-proteinase (BMP-1) inhibitor with IC50 of 44 nM, has excellent selectivity over MMPs.
More Information Supplier PageTAME 5mg | Purity Not Available
Selleck Chemicals
Idelalisib (CAL-101) 10mg | Purity Not Available
Selleck Chemicals
Idelalisib (CAL-101) is a selective p110δ inhibitor with IC50 of 2.5 nM in cell-free assays; shown to have 40- to 300-fold greater selectivity for p110δ than p110α/β/γ, and 400- to 4000-fold more selectivity to p110δ than C2β, hVPS34, DNA-PK and mTOR. Idelalisib also stimulates autophagy.
More Information Supplier PageIdelalisib (CAL-101) 50mg | Purity Not Available
Selleck Chemicals
Idelalisib (CAL-101) is a selective p110δ inhibitor with IC50 of 2.5 nM in cell-free assays; shown to have 40- to 300-fold greater selectivity for p110δ than p110α/β/γ, and 400- to 4000-fold more selectivity to p110δ than C2β, hVPS34, DNA-PK and mTOR. Idelalisib also stimulates autophagy.
More Information Supplier PageIdelalisib (CAL-101) 10mM/1mL | Purity Not Available
Selleck Chemicals
Idelalisib (CAL-101) is a selective p110δ inhibitor with IC50 of 2.5 nM in cell-free assays; shown to have 40- to 300-fold greater selectivity for p110δ than p110α/β/γ, and 400- to 4000-fold more selectivity to p110δ than C2β, hVPS34, DNA-PK and mTOR. Idelalisib also stimulates autophagy.
More Information Supplier PageBelnacasan (VX-765) 10mg | Purity Not Available
Selleck Chemicals
Belnacasan (VX-765) is a potent and selective inhibitor of caspase-1 with Ki of 0.8 nM in a cell-free assay. Phase 2.
More Information Supplier PageBelnacasan (VX-765) 50mg | Purity Not Available
Selleck Chemicals
Belnacasan (VX-765) is a potent and selective inhibitor of caspase-1 with Ki of 0.8 nM in a cell-free assay. Phase 2.
More Information Supplier PageGalunisertib (LY2157299) 5mg | Purity Not Available
Selleck Chemicals
Galunisertib (LY2157299) is a potent TGFβ receptor I (TβRI) inhibitor with IC50 of 56 nM in a cell-free assay. Phase 2/3.
More Information Supplier PageGalunisertib (LY2157299) 50mg | Purity Not Available
Selleck Chemicals
Galunisertib (LY2157299) is a potent TGFβ receptor I (TβRI) inhibitor with IC50 of 56 nM in a cell-free assay. Phase 2/3.
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