Darapladib 5mg | Purity Not Available
Selleck Chemicals
Darapladib is a reversible lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with IC50 of 0.25 nM. Phase 3.
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Darapladib 25mg | Purity Not Available
Selleck Chemicals
Darapladib is a reversible lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with IC50 of 0.25 nM. Phase 3.
More Information Supplier PageEntospletinib (GS-9973) 10mg | Purity Not Available
Selleck Chemicals
Entospletinib (GS-9973) is an orally bioavailable, selective Syk inhibitor with IC50 of 7.7 nM in a cell-free assay and showed 13- to >1000-fold cellular selectivity for Syk over other kinases(including Jak2, ckit, Flt3, Ret, KDR) as assessed by target protein phosphorylation or functional response.
More Information Supplier PageEntospletinib (GS-9973) 50mg | Purity Not Available
Selleck Chemicals
Entospletinib (GS-9973) is an orally bioavailable, selective Syk inhibitor with IC50 of 7.7 nM in a cell-free assay and showed 13- to >1000-fold cellular selectivity for Syk over other kinases(including Jak2, ckit, Flt3, Ret, KDR) as assessed by target protein phosphorylation or functional response.
More Information Supplier PageGNE-7915 50mg | Purity Not Available
Selleck Chemicals
GNE-7915 is a highly potent, selective, and brain-penetrable leucine-rich repeat kinase 2 (LRRK2) inhibitor, with IC50 and Ki of 9 nM and 1 nM, respectively.
More Information Supplier PageGNF-5 100mg | Purity Not Available
Selleck Chemicals
GNF-5 is a selective and allosteric Bcr-Abl inhibitor with IC50 of 220 nM.
More Information Supplier PageXMD8-92 50mg | Purity Not Available
Selleck Chemicals
XMD8-92 is a potent and selective dual inhibitor of big map kinase (BMK1, ERK5) and bromodomain-containing proteins (BRDs, BET) with Kd of 80 nM and 170 nM for ERK5 and BRD4(1), respectively.
More Information Supplier PageFR 180204 25mg | Purity Not Available
Selleck Chemicals
FR 180204 is an ATP-competitive, selective ERK inhibitor with Ki of 0.31 μM and 0.14 μM for ERK1 And ERK2, respectively. It is 30-fold less potent against the related kinase p38α and failed to inhibit any kinases(MEK1, MKK4, IKKα, PKCα, Src, Syc, and PDGFα) at less than 30 μM.
More Information Supplier PageEntospletinib (GS-9973) 200mg | Purity Not Available
Selleck Chemicals
Entospletinib (GS-9973) is an orally bioavailable, selective Syk inhibitor with IC50 of 7.7 nM in a cell-free assay and showed 13- to >1000-fold cellular selectivity for Syk over other kinases(including Jak2, ckit, Flt3, Ret, KDR) as assessed by target protein phosphorylation or functional response.
More Information Supplier PageHJC0350 50mg | Purity Not Available
Selleck Chemicals
HJC0350 is a potent and selective EPAC2 inhibitor with IC50 of 0.3 μM, exhibiting no inhibition on Epac1.
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