Selleck Chemicals
Epacadostat (INCB024360) analogue (INCB14943) is a potent, competitive IDO1 (indoleamine-(2,3)-dioxygenase) inhibitor with IC50 of 67 nM.
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Reversine
25mg
| Purity Not Available
Selleck Chemicals
Reversine is a potent human A3 adenosine receptor antagonist with Ki of 0.66 μM, and a pan-aurora A/B/C kinase inhibitor with IC50 of 400 nM/500 nM/400 nM, respectively. Also used for stem cell dedifferentiation.
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N6022
25mg
| Purity Not Available
Selleck Chemicals
N6022 is a selective, and reversible inhibitor of S-nitrosoglutathione reductase (GSNOR) with IC50 of 8 nM and Ki of 2.5 nM. Phase 1/2.
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BRD4770
25mg
| Purity Not Available
Selleck Chemicals
UNC0379
25mg
| Purity Not Available
Selleck Chemicals
UNC0379 is a selective, substrate competitive inhibitor of N-lysine methyltransferase SETD8 with IC50 of 7.3 μM, high selectivity over 15 other methyltransferases.
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LMK-235
200mg
| Purity Not Available
Selleck Chemicals
LMK-235
50mg
| Purity Not Available
Selleck Chemicals
LMK-235
10mg
| Purity Not Available
Selleck Chemicals
IM-12
50mg
| Purity Not Available
Selleck Chemicals
WH-4-023
25mg
| Purity Not Available
Selleck Chemicals
WH-4-023 (KIN001-112, KIN112, Dual LCK/SRC inhibitor) is a potent and orally active Lck/Src inhibitor withIC50s of 2 nM and 6 nM in cell-free assays, respectively. Exhibits >300-fold selectivity against p38α and KDR. Also potently inhibits SIK (IC50 values are 10, 22 and 60 nM for SIK 1, 2 and 3 respectively) and displays selectivity over […]
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