S1RA is a selective sigma-1 receptor antagonist, with a reported binding affinity of Ki = 17.0 ?? 7.0 nM, selective over the sigma-2 receptor and against a panel of other 170 receptors, enzymes, transporters and ion channels.
More Information Supplier PageS1RA is a selective sigma-1 receptor antagonist, with a reported binding affinity of Ki = 17.0 ?? 7.0 nM, selective over the sigma-2 receptor and against a panel of other 170 receptors, enzymes, transporters and ion channels.
More Information Supplier PageAlmorexant(ACT078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.
More Information Supplier PageAlmorexant(ACT078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.
More Information Supplier PageAlmorexant(ACT078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.
More Information Supplier PageABT-199 is a so-called BH3-mimetic drug, which is designed to block the function of the protein Bcl 2.
More Information Supplier PageABT-199 is a so-called BH3-mimetic drug, which is designed to block the function of the protein Bcl 2.
More Information Supplier PageABT-199 is a so-called BH3-mimetic drug, which is designed to block the function of the protein Bcl 2.
More Information Supplier PageABT-199 is a so-called BH3-mimetic drug, which is designed to block the function of the protein Bcl 2.
More Information Supplier PageVU 0361737 is a selective positive allosteric modulator at mGluR-4 (EC50 values are 240 and 110 nM at human and rat receptors respectively).
More Information Supplier Page
