Sotuletinib (BLZ945) is an orally active, potent and selective CSF-1R inhibitor with IC50 of 1 nM, >1000-fold selective against its closest receptor tyrosine kinase homologs.
More Information Supplier PageBikinin is an ATP-competitive Arabidopsis GSK-3 inhibitor, and acts as a strong activator of brassinosteroid (BR) signaling.
More Information Supplier PageSBE 13 HCl is a potent and selective PLK1 inhibitor with IC50 of 200 pM, >4000-fold selectivity over Aurora A kinase, Plk2 and Plk3.
More Information Supplier PageSBE 13 HCl is a potent and selective PLK1 inhibitor with IC50 of 200 pM, >4000-fold selectivity over Aurora A kinase, Plk2 and Plk3.
More Information Supplier PageCCG-1423 is a specific RhoA pathway inhibitor, which inhibits SRF-mediated transcription.
More Information Supplier PageCCG-1423 is a specific RhoA pathway inhibitor, which inhibits SRF-mediated transcription.
More Information Supplier PageBMH-21 is a DNA intercalator, which binds ribosomal DNA and inhibits RNA polymerase I (Pol I) transcription.
More Information Supplier PageYK-4-279 is a potent inhibitor of EWS-FLI1 binding to RNA helicase A (RHA).
More Information Supplier PageYK-4-279 is a potent inhibitor of EWS-FLI1 binding to RNA helicase A (RHA).
More Information Supplier PageSP2509 (HCI-2509) is a selective histone demethylase LSD1 inhibitor with IC50 of 13 nM, showing no activity against MAO-A, MAO-B, lactate dehydrogenase and glucose oxidase. SP2509 induces apoptosis and promotes autophagy.
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