A 438079 hydrochloride 100 mg | 100.00%
TargetMol
A 438079 hydrochloride (A-438079 HCl) is a potent and selective P2X7 receptor antagonist with pIC50 of 6.9.
More Information Supplier PageA 438079 hydrochloride (A-438079 HCl) is a potent and selective P2X7 receptor antagonist with pIC50 of 6.9.
More Information Supplier PageElacridar (GF120918) is an effective BCRP and P-gp (MDR-1) inhibitor.
More Information Supplier PageElacridar (GF120918) is an effective BCRP and P-gp (MDR-1) inhibitor.
More Information Supplier PageMK-8245 is a liver-targeting SCD inhibitor for human SCD1 (IC50: 1 nM) and for rat/mouse SCD1 (IC50: 3 nM), with anti-diabetic and anti-dyslipidemic function.
More Information Supplier PageMK-8245 is a liver-targeting SCD inhibitor for human SCD1 (IC50: 1 nM) and for rat/mouse SCD1 (IC50: 3 nM), with anti-diabetic and anti-dyslipidemic function.
More Information Supplier PageIDO5L (INCB024360 analogue) is an effective IDO1 inhibitor(IC50=10 nM).
More Information Supplier PageLY2784544(Gandotinib) is a potent JAK2 inhibitor (IC50: 3 nM), effective in JAK2V617F(Ki: 0.245 nM). The selectivity is higher 8- and 20-fold than JAK1 and JAK3.
More Information Supplier PageDecernotinib(VX-509; VRT-831509) is a potent and selective Janus kinase 3 (JAK3) inhibitor with Ki of 2.5 nM; IC50 is 50-170 nM in cellular assays.
More Information Supplier PageNSC319726, a mutant p53R175 reactivator, suppresses growth of fibroblasts that expresses the p53R175 mutation (IC50 = 8 nM).
More Information Supplier PageNSC319726, a mutant p53R175 reactivator, suppresses growth of fibroblasts that expresses the p53R175 mutation (IC50 = 8 nM).
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