TRPV1 antagonist 6 | MedChemExpress (MCE)

TRPV1 antagonist 6 (compound 51) is a mode-selective antagonist for transient receptor potential vanilloid member 1 (TRPV1), which shows antagonism with IC50 of 2.85 nM to capsaicin activation and 28.48 % inhibition against proton activation at a 3 µM concentration[1].

Trivial name TRPV1 antagonist 6
Catalog Number HY-161273
Research Area Neurological Disease
Purity ≥98.0%
SMILES CC(C)(C)C1=NN(C(CNC(NC2=CC=CC(N3CCO)=C2C=CC3=O)=O)=C1)C4=CC=CC(Cl)=C4
Size 1 mg
Supplier Page https://www.medchemexpress.com/trpv1-antagonist-6.html