Trimegestone-13C,d3 | MedChemExpress (MCE)
Trimegestone-13C,d3 is 13C and deuterated labeled Trimegestone (HY-106827). Trimegestone (RU 27987) is an orally active 19-norpregnane progestin. Trimegestone binds to progesterone receptor (PR) with an IC50 value of 3.3 nM (rat PR). Trimegestone increases alkaline phosphatase activity (EC50=0.1 nM) but not luciferase activity. Trimegestone also shows a weak antiandrogenic activity (weak androgen receptor affinity). Trimegestone can be used in studies of contraception or menopausal syndromes[1][2].
| Trivial name | Trimegestone-13C,d3 |
| Catalog Number | HY-106827S1 |
| Alternative Name(s) | RU 27987-13C,d3 |
| Research Area | Endocrinology |
| Purity | ≥98.0% |
| SMILES | C[C@@]12[C@](CC[C@]2(C)C([C@@H](O)[13C]([2H])([2H])[2H])=O)([H])[C@@]3([H])C(CC1)=C4C(CC3)=CC(CC4)=O |
| Size | 1 mg |
| Supplier Page | https://www.medchemexpress.com/trimegestone-13c-d3.html |