TEAD-IN-9 | MedChemExpress (MCE)

TEAD-IN-9 is a TEAD1 inhibitor with an IC50 of 0.29 μM. TEAD-IN-9 targets the palmitoyl pocket of TEAD, thereby effectively inhibiting the binding of YAP-TEAD and blocking the transcriptional function of YAP-TEAD (WO2024061366A1; compound 17)[1].

Trivial name TEAD-IN-9
Catalog Number HY-161443
Research Area Cancer
Purity ≥98.0%
SMILES O=P(C)(C)C1=CC=C(NCC2=CC=C(C(F)(F)F)C=C2)C(C3=NC(OC4COC4)=CC=N3)=C1
Size 1 mg
Supplier Page https://www.medchemexpress.com/tead-in-9.html