20S Proteasome-IN-5 | MedChemExpress (MCE)

20S Proteasome-IN-5 (Compound 5) is a macrocyclic inhibitor of the 20S Proteasome, with IC50 values of 0.19 and 52.5 μM for ChT-L and PGPH-L activity, respectively[1].

Trivial name 20S Proteasome-IN-5
Catalog Number HY-158150
Research Area Cancer
Purity ≥98.0%
SMILES CC(N[C@H](C(N[C@@H](CC(C)C)C(N[C@H](C(N[C@H](C([C@]1(CO1)C)=O)CC(C)C)=O)CC23)=O)=O)CC4=C(C([N+]([O-])=O)=CC=C4)OC5=CC3=C(C=C5)NC2=O)=O
Size 1 mg
Supplier Page https://www.medchemexpress.com/20s-proteasome-in-5.html