σ1 Receptor/μ Opioid receptor modulator 2 | MedChemExpress (MCE)
σ1 Receptor/μ Opioid receptor modulator 2 (compound 4x) is a dual μOR agonist/σ1R antagonist, and displays picomolar μOR agonism activity (EC50: 0.6 ± 0.2 nM) and good σ1R inhibitory activity (Ki: 363.7 ± 5.6 nM). σ1 Receptor/μ Opioid receptor modulator 2 exhibits robust analgesic effects in various pain models[1].
| Trivial name | σ1 Receptor/μ Opioid receptor modulator 2 |
| Catalog Number | HY-163065 |
| Research Area | Neurological Disease |
| Purity | ≥98.00% |
| SMILES | O=C(N(C1=CC=CC=N1)CC(N2CCC(CC2)C3=CC=CC=C3)CC)CC |
| PubChem Chemical Structure ID | 169494201 |
| Size | 1 mg |
| Supplier Page | https://www.medchemexpress.com/σ1-receptor-μ-opioid-receptor-modulator-2.html |