CRT0066101 | MedChemExpress (MCE)
CRT0066101 is a potent and orally active PKD inhibitor with IC50 values of 1 nM, 2.5 nM and 2 nM for PKD1, PKD2, and PKD3, respectively[1]. CRT0066101 is also a potent PIM2 inhibitor with an IC50 of ~135.7 nM. CRT0066101 has anticancer effects[2].
| Trivial name | CRT0066101 |
| Catalog Number | HY-15698 |
| Research Area | Cancer |
| CAS# | 956123-34-5 |
| Purity | ≥98.0% |
| SMILES | N[C@H](CC)CNC1=NC(C2=C(O)C=CC(C3=CN(C)N=C3)=C2)=NC=C1 |
| Size | 10 mg |
| Supplier Page | https://www.medchemexpress.com/crt0066101.html |