MS417
MS417 is a selective BET-specific BRD4 inhibitor, binds to BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively, with weak selectivity at CBP BRD (IC50, 32.7 μM).
| Trivial name | GTPL7512 |
| Catalog Number | S7615 |
| CAS# | 916489-36-6 |
| Size | 1g |
| Supplier Page | http://www.selleckchem.com/products/ms417.html |
| Additional Information | https://file.selleck.cn/downloads/struct/S7615-MS417-chemical-structure.png |