Rolapitant hydrochloride

Rolapitant (SCH619734) hydrochloride is a potent, selective, long-acting and orally active neurokinin 1 (NK1) receptor antagonist with a K i of 0.66 nM. Rolapitant hydrochloride does not interact with CYP3A4. Rolapitant hydrochloride shows potent centrally-mediated anti-emetic activity in both acute and delayed ferret emesis models [1] [2].

Price Not Available 100 mg Rolapitant hydrochloride Supplier Page

Catalog Number	T3724
Alternative Name(s)	Rolapitant HCl
Research Area	Neuroscience\|\|\|GPCR/G Protein
Molecular Formula	C25H27ClF6N2O2
CAS#	858102-79-1
Purity	98.46%
SMILES	Cl.C[C@@H](OC[C@]1(CC[C@]2(CCC(=O)N2)CN1)c1ccccc1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F
Size	100 mg
Supplier Page	https://www.targetmol.com/compound/Rolapitant hydrochloride
Additional Information	https://www.targetmol.com/datasheet/T3724