Pitolisant hydrochloride
Pitolisant (Tiprolisant, BF-2649) acts as a high-affinity competitive antagonist (Ki=0.16 nM) and as an inverse agonist (EC50=1.5 nM) at the human histamine H3 receptor subtype.
Trivial name | Tiprolisant hydrochloride, BF-2649 HCl |
Catalog Number | S5926 |
Molecular Formula | C17H27Cl2NO |
CAS# | 903576-44-3 |
Inchi | InChI=1S/C17H26ClNO.ClH/c18-17-9-7-16(8-10-17)6-4-14-20-15-5-13-19-11-2-1-3-12-19;/h7-10H,1-6,11-15H2;1H |
Inchi Key | XLFKECRRMPOAQS-UHFFFAOYSA-N |
SMILES | C1CCN(CC1)CCCOCCCC2=CC=C(C=C2)Cl.Cl |
Size | 25mg |
Supplier Page | http://www.selleckchem.com/products/pitolisant-hydrochloride.html |
Additional Information | https://file.selleck.cn/downloads/struct/pitolisant-hydrochloride-chemical-structure-s5926.gif |