GSK 5959
GSK5959 is a potent and selective BRPF1 bromodomain inhibitor with an IC50 of 80 nM and exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.
| Trivial name | N/A |
| Catalog Number | S5916 |
| Molecular Formula | C22H26N4O3 |
| CAS# | 901245-65-6 |
| Inchi | InChI=1S/C22H26N4O3/c1-24-18-13-16(23-21(27)15-9-5-6-10-20(15)29-3)17(26-11-7-4-8-12-26)14-19(18)25(2)22(24)28/h5-6,9-10,13-14H,4,7-8,11-12H2,1-3H3,(H,23,27) |
| Inchi Key | LTUGYAOMCKNTGG-UHFFFAOYSA-N |
| SMILES | CN1C2=C(C=C(C(=C2)NC(=O)C3=CC=CC=C3OC)N4CCCCC4)N(C1=O)C |
| Size | 25mg |
| Supplier Page | http://www.selleckchem.com/products/gsk-5959.html |
| Additional Information | https://file.selleck.cn/downloads/struct/gsk-5959-chemical-structure-s5916.gif |