Dabigatran etexilate mesylate
Dabigatran etexilate mesylate (Pradaxa, BIBR 1048MS, Dabigatran etexilate methanesulfonate) is an orally active prodrug of Dabigatran which is a reversible and selective, direct thrombin inhibitor (DTI). Dabigatran selectively and reversibly inhibits human thrombin with Ki of 4.5 nM and thrombin-induced platelet aggregation with IC50 of 10 nM.
Trivial name | Pradaxa, BIBR 1048MS, Dabigatran etexilate methanesulfonate |
Catalog Number | S5960 |
Molecular Formula | C35H45N7O8S |
CAS# | 872728-81-9 |
Inchi | #N/A |
Inchi Key | #N/A |
SMILES | CCCCCCOC(=O)NC(=N)C1=CC=C(NCC2=NC3=C(C=CC(=C3)C(=O)N(CCC(=O)OCC)C4=CC=CC=N4)[N]2C)C=C1.C[S](O)(=O)=O |
Size | 100mg |
Supplier Page | http://www.selleckchem.com/products/dabigatran-etexilate-mesylate.html |
Additional Information | https://file.selleck.cn/downloads/struct/s5960-dabigatran-etexilate-mesylate-chemical-structure.gif |