BPTU
Allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM). Non-nucleotide ligand. Binds receptor outside of the helical bundle. Blocks inhibition of spontaneous contraction of rat and mouse colon induced by electrical field stimulation, nicotine and P2Y agonists. Antithrombotic; reduces platelet aggregation.
| Catalog Number | T4132 |
| Alternative Name(s) | BMS-646786 |
| Research Area | GPCR/G Protein|||Neuroscience |
| Molecular Formula | C23H22F3N3O3 |
| CAS# | 870544-59-5 |
| Purity | 99.89% |
| SMILES | CC(C)(C)C1=CC=CC=C1OC2=C(C=CC=N2)NC(=O)NC3=CC=C(C=C3)OC(F)(F)F |
| Size | 5 mg |
| Supplier Page | https://www.targetmol.com/compound/BPTU |
| Additional Information | https://www.targetmol.com/datasheet/T4132 |