Nelotanserin
Nelotanserin is a potent 5-HT2A inverse agonist, a moderately potent 5-HT2C partial inverse agonist and a weak 5-HT2B inverse agonist, with IC50s of 1.7, 79, 791 nM in IP accumulation assays, respectively.
Trivial name | APD125 |
Catalog Number | E7981 |
Molecular Formula | C22H19N5O |
CAS# | 839713-36-9 |
Inchi | InChI=1S/C22H19N5O/c1-13-4-2-5-18(25-13)21-20(19-6-3-11-27(19)26-21)15-9-10-24-17-8-7-14(22(23)28)12-16(15)17/h2,4-5,7-10,12H,3,6,11H2,1H3,(H2,23,28) |
Inchi Key | IVRXNBXKWIJUQB-UHFFFAOYSA-N |
SMILES | CC1=NC(=CC=C1)C2=NN3CCCC3=C2C4=C5C=C(C=CC5=NC=C4)C(=O)N |
Size | 5mg |
Supplier Page | http://www.selleckchem.com/products/nelotanserin.html |
Additional Information | https://file.selleck.cn/downloads/struct/e7981-nelotanserin-chemical-structure-tube.png |