WDR5-0102
WDR5-0102 is an inhibitor targeting WDR5-MLL1 interface (K dis =7 μM, K d =4 μM). WDR5-0102 suppresses MLL1 HMT activity, but not human H3K4 methyltransferase SETD7 and six other HMTs: G9a, EHMT1, SUV39H2, SETD8, PRMT3 , and PRMT5 .
| Catalog Number | T67947 |
| Research Area | Chromatin/Epigenetic |
| Molecular Formula | C18H19ClN4O3 |
| CAS# | 824960-50-1 |
| Purity | 97.16% |
| SMILES | O=C(NC1=CC(=CC=C1N2CCN(C)CC2)N(=O)=O)C=3C=CC=CC3Cl |
| Size | 1 mL |
| Supplier Page | https://www.targetmol.com/compound/wdr5-0102 |
| Additional Information | https://www.targetmol.com/datasheet/T67947 |