WDR5-0102| ChemScene
WDR5-0102 is an inhibitor targeting WDR5-MLL1 interface (Kdis=7 μM, Kd=4 μM). WDR5-0102 suppresses MLL1 HMT activity, but not human H3K4 methyltransferase SETD7 and six other HMTs: G9a, EHMT1, SUV39H2, SETD8, PRMT3, and PRMT5[2].
| Trivial name | WDR5-0102 |
| Catalog Number | CS-0641680 |
| Molecular Formula | 374.82 |
| CAS# | 824960-50-1 |
| Purity | >98% |
| Condensed Formula | C18H19ClN4O3 |
| Size | 50mg |
| Supplier Page | www.chemscene.com/824960-50-1.html |