GSK180736A (GSK180736)

GSK180736A (GSK180736), developed as a Rho-associated, coiled-coil-containing protein kinase inhibitor, binds to GRK2(G protein-coupled receptor kinase 2) with logIC50 pf -6.6 (logIC50 -4.0 for GRK5 and >-3 for GRK1); ≥400-fold selective for GRK2 over both GRK1 and GRK5.

Price Not Available 10mg GSK180736A (GSK180736) Supplier Page

Trivial name	N/A
Catalog Number	S8489
Molecular Formula	C19H16FN5O2
CAS#	817194-38-0
Inchi	InChI=1S/C19H16FN5O2/c1-10-16(17(24-19(27)22-10)11-2-4-13(20)5-3-11)18(26)23-14-6-7-15-12(8-14)9-21-25-15/h2-9,17H,1H3,(H,21,25)(H,23,26)(H2,22,24,27)
Inchi Key	HEAIGWIZTYAQTC-UHFFFAOYSA-N
SMILES	CC1=C(C(NC(=O)N1)C2=CC=C(C=C2)F)C(=O)NC3=CC4=C(C=C3)NN=C4
Size	10mg
Supplier Page	http://www.selleckchem.com/products/gsk180736a.html
Additional Information	https://file.selleck.cn/downloads/struct/gsk180736a-chemical-structure-S8489.gif