(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

Selective vasopressin V1A receptor antagonist. Inhibits vasopressin and oxytocin-induced increases in intracellular calcium concentrations in vitro (IC50 values are 5 and 30 nM respectively). Exhibits potent and prolonged antivasopressor activity and induces anxiolytic-like effects in the dorsal, but not ventral, hippocampus in vivo.

Catalog Number TP2136
Molecular Formula C52H74N14O12S2
CAS# 73168-24-8
Size 10 mg
Supplier Page https://www.targetmol.com/compound/(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
Additional Information https://www.targetmol.com/datasheet/TP2136