(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
Selective vasopressin V1A receptor antagonist. Inhibits vasopressin and oxytocin-induced increases in intracellular calcium concentrations in vitro (IC50 values are 5 and 30 nM respectively). Exhibits potent and prolonged antivasopressor activity and induces anxiolytic-like effects in the dorsal, but not ventral, hippocampus in vivo.
Catalog Number | TP2136 |
Molecular Formula | C52H74N14O12S2 |
CAS# | 73168-24-8 |
Size | 10 mg |
Supplier Page | https://www.targetmol.com/compound/(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin |
Additional Information | https://www.targetmol.com/datasheet/TP2136 |