phentolamine hydrochloride

Phentolamine hydrochloride is a potent, selective, and orally active antagonist of α1 and α2 adrenergic receptors , with pKi values of 8.8, 8.0, and 8.3 for the human α2A, α2B, and α2C adrenergic receptors, respectively. It also shows binding affinities for the α1-adrenoceptor subtypes, exhibiting Ki values of 6.1 nM for cloned α1A/D, 39.8 nM for α1B, and 2.8 nM for α1C.

Price Not Available 5mg phentolamine hydrochloride Supplier Page

Catalog Number	E6046
Molecular Formula	C16H17Cl2N5O2
CAS#	73-05-2
Inchi	InChI=1S/C16H17Cl2N5O2/c17-10-2-1-3-11(18)13(10)15(24)22-12-8-20-23-14(12)16(25)21-9-4-6-19-7-5-9/h1-3,8-9,19H,4-7H2,(H,20,23)(H,21,25)(H,22,24)
Inchi Key	OVPNQJVDAFNBDN-UHFFFAOYSA-N
SMILES	C1CNCCC1NC(=O)C2=C(C=NN2)NC(=O)C3=C(C=CC=C3Cl)Cl
Size	5mg
Supplier Page	http://www.selleckchem.com/products/phentolamine-hydrochloride.html
Additional Information	https://file.selleck.cn/downloads/struct/E6046-phentolamine-hydrochloride-chemical-structure.png