Elacestrant
Elacestrant (RAD1901) is an orally available and selective estrogen receptor degrader (SERD) with IC50s of 48 and 870 nM for ERα and ERβ, respectively. Elacestrant also can inhibit growth of ER+ breast cancer cell lines in vitro and in vivo.
| Trivial name | RAD191 |
| Catalog Number | E7121 |
| Molecular Formula | C10H20N2S4 |
| CAS# | 722533-56-4 |
| Inchi | InChI=1S/C10H20N2S4/c1-5-11(6-2)9(13)15-16-10(14)12(7-3)8-4/h5-8H2,1-4H3 |
| Inchi Key | AUZONCFQVSMFAP-UHFFFAOYSA-N |
| SMILES | CCN(CC)C(=S)SSC(=S)N(CC)CC |
| Size | 1mg |
| Supplier Page | http://www.selleckchem.com/products/elacestrant-e7121.html |
| Additional Information | https://file.selleck.cn/downloads/struct/e7121-elacestrant-chemical-structure-tube.png |