Astemizole 100mg

Astemizole is a potent antihistamine (H1-receptor antagonist, IC50 = 4 nM) that displays selectivity over dopamine, 5-HT, and muscarinic acetylcholine receptors. This compound has shown potent hERG K+ channel blocking activity (IC50 = 0.9 nM), antimalarial activity in multidrug resistant strains in vitro (IC50 = 227 – 734 nM), and has been used as a chaperone to correct folding defects and restore protein function for some mutated forms of hERG channels.

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Trivial name Astemizole 100mg
Catalog Number A13899-100
Alternative Name(s) 1-[(4-Fluorophenyl)methyl]-N-[1-[2-(4-methoxyphenyl)ethyl]-4-piperidinyl]-1H-benzimidazol-2-amine
Molecular Formula C28H31FN4O
CAS# 68844-77-9
SMILES COC1=CC=C(C=C1)CCN2CCC(CC2)NC3=NC4=CC=CC=C4N3CC5=CC=C(C=C5)F
Size 100mg
Supplier Page http://www.adooq.com/astemizole.html