Pimethixene
Pimethixene(Calmixen, Pimetixene) is a highly potent and non-selective antagonist of the 5-HT2B receptor, with a pKi of 10.44. It also functions as an antihistamine and anticholinergic agent, and is a highly potent multi-target antagonist with antagonistic effects on multiple receptors.
Trivial name | Calmixen, Pimetixene |
Catalog Number | E4862 |
Molecular Formula | C28H24FN3O5 |
CAS# | 314-03-4 |
Inchi | InChI=1S/C28H24FN3O5/c1-35-24-15-21-22(16-25(24)36-2)30-14-11-23(21)37-20-9-7-19(8-10-20)32-27(34)28(12-13-28)26(33)31-18-5-3-17(29)4-6-18/h3-11,14-16H,12-13H2,1-2H3,(H,31,33)(H,32,34) |
Inchi Key | ONIQOQHATWINJY-UHFFFAOYSA-N |
SMILES | COC1=CC2=C(C=CN=C2C=C1OC)OC3=CC=C(C=C3)NC(=O)C4(CC4)C(=O)NC5=CC=C(C=C5)F |
Size | 100mg |
Supplier Page | http://www.selleckchem.com/products/pimethixene.html |
Additional Information | https://file.selleck.cn/downloads/struct/E4862-Pimethixene-chemical-structure.png |