LMTK3-IN-1 | MedChemExpress (MCE)
LMTK3-IN-1 (compound C28) is an ATP-competitive inhibitor of lemur tyrosine kinase 3 (LMTK3) (Kd=2.5 μM)，that acts by degrading LMTK3 via the ubiquitin-proteasome pathway. LMTK3-IN-1 shows anticancer activity in a variety of cancer cell lines and in vivo BC mouse models. LMTK3-IN-1 induces apoptosis in BC cell lines at 10-20 μM[1].
| Trivial name | LMTK3-IN-1 |
| Catalog Number | HY-153896 |
| Research Area | Cancer |
| CAS# | 2764850-23-7 |
| Purity | 98.74% |
| SMILES | FC(F)(OC1=CC=CC(C2=CN=C3C=CC(C4=CC=NC=C4)=NN32)=C1)F |
| PubChem Chemical Structure ID | 138454301 |
| Size | 5 mg |
| Supplier Page | https://www.medchemexpress.com/lmtk3-in-1.html |