CDK12-IN-4

CDK12-IN-4, a pyrazolotriazine compound, exhibits potent inhibition of CDK12 by achieving an IC50 value of 0.641 μM, utilizing high ATP levels (2 mM). Notably, CDK12-IN-4 does not impact CDK2/Cyclin E (IC50 > 20 μM) or CDK9/Cyclin T1 (IC50 > 20 μM) under the influence of high ATP (2 mM) levels (WO2021116178A1).

Price Not Available 5 mg CDK12-IN-4 Supplier Page

Catalog Number	T40288
Alternative Name(s)	CDK12-IN-4
Molecular Formula	C20H20F2N8O
CAS#	2651196-69-7
SMILES	Fc1ccc2nc(CNc3nc(nc4c(cnn34)C3CC3)N3CCOCC3)[nH]c2c1F
Size	5 mg
Supplier Page	https://www.targetmol.com/compound/cdk12-in-4
Additional Information	https://www.targetmol.com/datasheet/T40288