BBC0403
BBC0403 is a small-molecule selective inhibitor of Bromodomain-containing protein 2(BRD2) with Kds of 7.64 μM and 41.37 μM for BRD2 (BD2) and BRD2 (BD1), respectively. It is a potential intra-articular injectable therapeutic agent for treating osteoarthritis (OA).
| Catalog Number | E4713 |
| Molecular Formula | C26H29Cl2N5O3 |
| CAS# | 2644662-83-7 |
| Inchi | InChI=1S/C26H29Cl2N5O3/c1-32-6-8-33(9-7-32)5-4-10-36-25-13-21-18(11-24(25)35-3)26(17(15-29)16-30-21)31-22-14-23(34-2)20(28)12-19(22)27/h11-14,16H,4-10H2,1-3H3,(H,30,31) |
| Inchi Key | UBPYILGKFZZVDX-UHFFFAOYSA-N |
| SMILES | CN1CCN(CC1)CCCOC2=C(C=C3C(=C2)N=CC(=C3NC4=CC(=C(C=C4Cl)Cl)OC)C#N)OC |
| Size | 5mg |
| Supplier Page | http://www.selleckchem.com/products/bbc0403.html |
| Additional Information | https://file.selleck.cn/downloads/struct/E4713-BBC0403-chemical-structure.png |