Pelitinib (EKB-569)

Pelitinib (EKB-569) is a potent irreversible EGFR inhibitor with IC50 of 38.5 nM. Pelitinib (EKB-569) also slightly inhibits Src, MEK/ERK and ErbB2 with IC50s of 282 nM, 800 nM and 1255 nM, respectively. Phase2.

Price Not Available 5mg Pelitinib (EKB-569) Supplier Page
Trivial name N/A
Catalog Number S1392
Molecular Formula C20H23ClFNO
CAS# 257933-82-7
Inchi InChI=1S/C20H23ClFNO/c21-18-5-3-17(4-6-18)20(24)14-23-11-9-16(10-12-23)13-15-1-7-19(22)8-2-15/h1-8,16,20,24H,9-14H2
Inchi Key GGUSQTSTQSHJAH-UHFFFAOYSA-N
SMILES C1CN(CCC1CC2=CC=C(C=C2)F)CC(C3=CC=C(C=C3)Cl)O
Size 5mg
Supplier Page http://www.selleckchem.com/products/Pelitinib.html
Additional Information https://file.selleck.cn/downloads/struct/Pelitinib-EKB-569-chemical-structure-S1392.gif