CPI-1612
CPI-1612 is a highly potent, orally active inhibitor of EP300/CBP histone acetyltransferase (HAT). It displays an IC50 of 8.0 nM for EP300 HAT. CPI-1612 suppresses H3K27 acetylation in vivo and exhibits efficacy in JEKO-1 mantle cell lymphoma xenograft at a low dose. CPI-1612 displays anticancer activity.
| Catalog Number | S6876 |
| CAS# | 2374971-81-8 |
| Size | 5mg |
| Supplier Page | http://www.selleckchem.com/products/cpi-1612.html |
| Additional Information | https://file.selleck.cn/downloads/struct/S6876-CPI-1612-chemical-structure.png |