uPSEM792 | MedChemExpress (MCE)
uPSEM792 is a pharmacologically selective effector molecules (PSEM) agonist for PSAM4-GlyR, with an affinity of Ki of 0.7 nM. uPSEM792 is a substrate for efflux transporters in brains of wild type and dual P-gp and BCRP knockout mice. uPSEM7952 is a possible lead for developing the PET radioligand for PSAM4-GlyR[1].
| Trivial name | uPSEM792 |
| Catalog Number | HY-161246 |
| Research Area | Neurological Disease |
| CAS# | 2323525-19-3 |
| Purity | ≥98.0% |
| SMILES | CN1C2=C(C=C(C3CNCC4C3)C4=C2)N=CC1=O |
| Size | 1 mg |
| Supplier Page | https://www.medchemexpress.com/upsem792.html |