ARV-471
A PROTAC that drives ER degradation
| Catalog Number | 43002 |
| Alternative Name(s) | Vepdegestrant |
| Research Area | Product Type|Biochemicals|PROTACs||Research Area|Cancer||Research Area|Cell Biology|Proteolysis|Ubiquitin/Proteasome System||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Estrogens & Progestins |
| Molecular Formula | C45H49N5O4 |
| CAS# | 2229711-68-4 |
| Purity | ≥98% |
| Inchi | InChI=1S/C45H49N5O4/c51-37-12-15-39-33(27-37)8-13-38(31-4-2-1-3-5-31)43(39)32-6-9-35(10-7-32)48-20-18-30(19-21-48)28-47-22-24-49(25-23-47)36-11-14-40-34(26-36)29-50(45(40)54)41-16-17-42(52)46-44(41)53/h1-7,9-12,14-15,26-27,30,38,41,43,51H,8,13,16-25,28-29H2,(H,46,52,53)/t38-,41+,43+/m1/s1 |
| Inchi Key | TZZDVPMABRWKIZ-XMOGEVODSA-N |
| SMILES | OC1=CC=C2[C@@H](C3=CC=C(N(CC4)CCC4CN5CCN(C6=CC=C7C(CN([C@@H](CCC8=O)C(N8)=O)C7=O)=C6)CC5)C=C3)[C@@H](C9=CC=CC=C9)CCC2=C1 |
| Size | 5 mg |
| Supplier Page | https://www.caymanchem.com/product/43002 |