MS1943
MS1943 is an orally bioavailable EZH2 selective degrader that effectively reduces EZH2 levels in cells with IC50 of 120 nM for inhibiting EZH2 methyltransferase activity.
| Trivial name | N/A |
| Catalog Number | S8918 |
| Molecular Formula | C42H54N8O3 |
| CAS# | 2225938-17-8 |
| SMILES | CC1=CC(=C(C(=O)N1)CNC(=O)C2=C3C=NN(C3=CC(=C2)C4=CN=C(C=C4)N5CCN(CC5)CCNC(=O)CC67CC8CC(C6)CC(C8)C7)C(C)C)C |
| Size | 1g |
| Supplier Page | http://www.selleckchem.com/products/ms1943.html |
| Additional Information | https://file.selleck.cn/downloads/struct/s8918-ms1943-chemical-structure.gif |