RK-287107
RK-287107 is a novel, potent and selective tankyrase inhibitor with antitumor activity. RK-287107 inhibits tankyrase-1 and tankyrase-2 in vitro with IC50 of 14.3 nM and 10.6 nM.
| Trivial name | N/A |
| Catalog Number | S8876 |
| Molecular Formula | C22H26F2N4O2 |
| CAS# | 2171386-10-8 |
| Inchi | InChI=1S/C22H26F2N4O2/c23-14-11-16(24)19-18(12-14)28(9-10-29)13-22(19)5-7-27(8-6-22)21-25-17-4-2-1-3-15(17)20(30)26-21/h11-12,29H,1-10,13H2,(H,25,26,30) |
| Inchi Key | FZQYCOUBRJEYBC-UHFFFAOYSA-N |
| SMILES | C1CCC2=C(C1)C(=O)NC(=N2)N3CCC4(CC3)CN(C5=C4C(=CC(=C5)F)F)CCO |
| Size | 5mg |
| Supplier Page | http://www.selleckchem.com/products/pk-287107.html |
| Additional Information | https://file.selleck.cn/downloads/struct/rk-287107-chemical-structure-s8876.gif |