Amcenestrant (SAR439859)
Amcenestrant (SAR439859, compound 43d) is an orally available and nonsteroidal selective estrogen receptor degrader (SERD) with potential antineoplastic activity. SAR439859 is a potent estrogen receptor (ER) antagonist with EC50 of 0.2 nM for ERα degradation.
Trivial name | N/A |
Catalog Number | S9609 |
Molecular Formula | C31H30Cl2FNO3 |
CAS# | 2114339-57-8 |
SMILES | C1CC2=C(C=CC(=C2)C(=O)O)C(=C(C1)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)OC5CCN(C5)CCCF |
Size | 25mg |
Supplier Page | http://www.selleckchem.com/products/sar439859.html |
Additional Information | https://file.selleck.cn/downloads/struct/s9609-sar439859-chemical-structure.gif |