ABCG2-IN-3 | MedChemExpress (MCE)

ABCG2-IN-3 (Compound 52) is a selective inhibitor for breast cancer resistance protein (ABCG2), with an IC50 of 0.238 µM. ABCG2-IN-3 reverses the ABCG2-mediated resistance toward SN-38 and inhibit the ATPase activity[1].

Trivial name ABCG2-IN-3
Catalog Number HY-119724
Research Area Cancer
CAS# 1942919-63-2
Purity ≥98.0%
SMILES COC1=CC=C(C=C1)C(N2C(C3=C(CC2)C(C=CC=C4)=C4N3)C5=CC(Cl)=C(C=C5)Cl)=O
Size 1 mg
Supplier Page https://www.medchemexpress.com/abcg2-in-3.html