GSK6853
GSK6853 is a selective benzimidazolone BRPF1 inhibitor with pIC50 of 8.1(TR-FRET) showing greater than 1600-fold selectivity over all other bromodomains tested.
| Trivial name | N/A |
| Catalog Number | S8265 |
| Molecular Formula | C22H27N5O3 |
| CAS# | 1910124-24-1 |
| Inchi | InChI=1S/C22H27N5O3/c1-14-13-23-9-10-27(14)17-12-19-18(25(2)22(29)26(19)3)11-16(17)24-21(28)15-7-5-6-8-20(15)30-4/h5-8,11-12,14,23H,9-10,13H2,1-4H3,(H,24,28)/t14-/m1/s1 |
| Inchi Key | FQWDVNSBYDXPIO-CQSZACIVSA-N |
| SMILES | CC1CNCCN1C2=CC3=C(C=C2NC(=O)C4=CC=CC=C4OC)N(C(=O)N3C)C |
| Size | 5mg |
| Supplier Page | http://www.selleckchem.com/products/gsk6853.html |
| Additional Information | https://file.selleck.cn/downloads/struct/gsk6853-chemical-structure-S8265.gif |