ARV-825
ARV-825 is a PROTAC targeting on BRD4, consisting of a BRD4-ligand JQ-1 linked to a cereblon E3 ligase ligand Pomalidomide, with Kds values of 90nM and 28nM for affinity to BD1 and BD2.
| Trivial name | / |
| Catalog Number | CSN18046 |
| Alternative Name(s) | / |
| Research Area | Cancer |
| Molecular Formula | C46H47ClN8O9S |
| CAS# | 1818885-28-7 |
| Purity | ≥98% |
| SMILES | CC1=NN=C2N1C(SC(C)=C3C)=C3C(C4=CC=C(Cl)C=C4)=N[C@H]2CC(NC5=CC=C(OCCOCCOCCOCCNC6=C(C(N(C7CCC(NC7=O)=O)C8=O)=O)C8=CC=C6)C=C5)=O |
| Size | 5mg |
| Supplier Page | https://www.csnpharm.com/products/arv-825.html |