GSK864
GSK864 is a cell-penetrant, potent, and selective inhibitor of isocitrate dehydrogenase 1 (IDH1) mutants, specifically targeting the R132C, R132H, and R132G variants with IC50 values of 8.8 nM, 15.2 nM, and 16.6 nM, respectively.
Catalog Number | S7994 |
CAS# | 1816331-66-4 |
Size | 1g |
Supplier Page | http://www.selleckchem.com/products/gsk864.html |
Additional Information | https://file.selleck.cn/downloads/struct/S7994-GSK864-chemical-structure.png |