BIX-01294 hydrochloride hydrate | MedChemExpress (MCE)

BIX-01294 hydrochloride hydrate is a histone-lysine methyltransferase (HMTase) inhibitor, which selective inhibits the G9aHMTase with IC50 of 1.7 μM, reduces histone-3 lysine (9) methylation (H3K9me), induces autophagy and apoptosis in human glioma cells[1][2].

Trivial name BIX-01294 hydrochloride hydrate
Catalog Number HY-10587A
Research Area Cancer
CAS# 1808255-64-2
Purity ≥98.0%
SMILES COC1=CC2=C(NC3CCN(CC3)CC4=CC=CC=C4)N=C(N5CCN(CCC5)C)N=C2C=C1OC.Cl.O.Cl.Cl.[x]
Size 1 mg
Supplier Page https://www.medchemexpress.com/bix-01294-hydrochloride-hydrate.html