Enzastaurin
Enzastaurin is a potent PKCβ selective inhibitor with IC50 of 6 nM in cell-free assays, 6- to 20-fold selectivity against PKCα, PKCγ and PKCε. Phase 3.
Trivial name | LY317615 |
Catalog Number | S1055 |
Molecular Formula | C32H29N5O2 |
CAS# | 170364-57-5 |
Inchi | InChI=1S/C32H29N5O2/c1-35-19-25(23-9-2-4-11-27(23)35)29-30(32(39)34-31(29)38)26-20-37(28-12-5-3-10-24(26)28)22-13-16-36(17-14-22)18-21-8-6-7-15-33-21/h2-12,15,19-20,22H,13-14,16-18H2,1H3,(H,34,38,39) |
Inchi Key | AXRCEOKUDYDWLF-UHFFFAOYSA-N |
SMILES | CN1C=C(C2=CC=CC=C21)C3=C(C(=O)NC3=O)C4=CN(C5=CC=CC=C54)C6CCN(CC6)CC7=CC=CC=N7 |
Size | 50mg |
Supplier Page | http://www.selleckchem.com/products/Enzastaurin.html |
Additional Information | https://file.selleck.cn/downloads/struct/Enzastaurin-LY317615-chemical-structure-S1055.gif |