Rimonabant (SR141716)
Rimonabant (SR141716) is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane. Rimonabant is also a dual inhibitor of acyl CoA:cholesterol acyltransferases(ACAT) 1 and 2 and inhibits mycobacterial MmpL3.
Trivial name | N/A |
Catalog Number | S3021 |
Molecular Formula | C22H21Cl3N4O |
CAS# | 168273-06-1 |
Inchi | InChI=1S/C22H21Cl3N4O/c1-14-20(22(30)27-28-11-3-2-4-12-28)26-29(19-10-9-17(24)13-18(19)25)21(14)15-5-7-16(23)8-6-15/h5-10,13H,2-4,11-12H2,1H3,(H,27,30) |
Inchi Key | JZCPYUJPEARBJL-UHFFFAOYSA-N |
SMILES | CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)Cl |
Size | 1g |
Supplier Page | http://www.selleckchem.com/products/rimonabant-sr141716.html |
Additional Information | https://file.selleck.cn/downloads/struct/Rimonabant-chemical-structure-s3021.gif |