GSK467

GSK467 is a cell penetrant and selective inhibitor of KDM5B (JARID1B/PLU1) with Ki of 10 nM. GSK467 shows apparent 180-fold selectivity for KDM4C and no measurable inhibitory effects toward KDM6 or other JmJ family members.

Price Not Available 5mg GSK467 Supplier Page
Trivial name N/A
Catalog Number S0269
Molecular Formula C17H13N5O2
CAS# 1628332-52-4
Inchi InChI=1S/C17H13N5O2/c23-16-14-6-7-18-9-15(14)20-17(21-16)24-13-8-19-22(11-13)10-12-4-2-1-3-5-12/h1-9,11H,10H2,(H,20,21,23)
Inchi Key ZTYRLXUTLYBVHH-UHFFFAOYSA-N
SMILES C1=CC=C(C=C1)CN2C=C(C=N2)OC3=NC4=C(C=CN=C4)C(=O)N3
Size 5mg
Supplier Page http://www.selleckchem.com/products/gsk467.html
Additional Information https://file.selleck.cn/downloads/struct/gsk467-chemical-structure-s0269.gif