Relacorilant | MedChemExpress (MCE)
Relacorilant is a potent, selective and orally bioavailable glucocorticoid receptor antagonist, with a Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively. Relacorilant has the potential for Cushing’s syndrome treatment.
| Trivial name | Relacorilant |
| Catalog Number | HY-109042 |
| Alternative Name(s) | CORT 125134 |
| Research Area | Endocrinology; Cardiovascular Disease |
| CAS# | 1496510-51-0 |
| Purity | 99.4% |
| SMILES | O=C(C1=CC(C(F)(F)F)=CC=N1)[C@@]2(CN(S(=O)(C3=CN(C)N=C3)=O)CC4)C4=CC5=C(C=NN5C6=CC=C(F)C=C6)C2 |
| Size | 50 mg |
| Supplier Page | https://www.medchemexpress.com/Relacorilant.html |