Tegaserod
Tegaserod is an orally active agonist of serotonin receptor 4 (5-HT4R) and also acts as an antagonist of 5-HT2B receptor with pKi values of 7.5, 8.4, and 7.0 for human recombinant 5-HT2A, 5-HT2B, and 5-HT2C receptors, respectively. Tegaserod has anti-tumor activity and is used in the research of irritable bowel syndrome (IBS).
Catalog Number | E4976 |
Molecular Formula | C6H12N2O4Pt |
CAS# | 145158-71-0 |
Inchi | InChI=1S/C6H8O4.2H3N.Pt/c7-4(8)6(5(9)10)2-1-3-6;;;/h1-3H2,(H,7,8)(H,9,10);2*1H3;/q;;;+2/p-2 |
Inchi Key | OLESAACUTLOWQZ-UHFFFAOYSA-L |
SMILES | C1CC(C1)(C(=O)O)C(=O)O.[NH2-].[NH2-].[Pt+2] |
Size | 5mg |
Supplier Page | http://www.selleckchem.com/products/tegaserod.html |
Additional Information | https://file.selleck.cn/downloads/struct/E4976-Tegaserod-chemical-structure.png |