Mozavaptan (hydrochloride)
Mozavaptan hydrochloride(OPC 31260 HCl), a benzazepine derivative is a potent, selective, competitive, and orally active antagonist of vasopressin V2 receptor with an IC50 value of 14 nM. Mozavaptan hydrochloride shows ~85-fold selectivity for V2 receptor over V1 receptor. Mozavaptan hydrochloride has the potential for hyponatremia, syndrome of inappropriate antidiuretic hormone (SIADH), and congestive heart failure treatment.
Trivial name | OPC 31260 HCl |
Catalog Number | E4957 |
Molecular Formula | C13H16N2O2 |
CAS# | 138470-70-9 |
Inchi | InChI=1S/C13H16N2O2/c1-9(16)14-6-5-10-8-15-13-4-3-11(17-2)7-12(10)13/h3-4,7-8,15H,5-6H2,1-2H3,(H,14,16) |
Inchi Key | DRLFMBDRBRZALE-UHFFFAOYSA-N |
SMILES | CC(=O)NCCC1=CNC2=C1C=C(C=C2)OC |
Size | 5mg |
Supplier Page | http://www.selleckchem.com/products/mozavaptan-hydrochloride.html |
Additional Information | https://file.selleck.cn/downloads/struct/E4957-Mozavaptan-hydrochloride-chemical-structure.png |