Mozavaptan (hydrochloride)

Mozavaptan hydrochloride(OPC 31260 HCl), a benzazepine derivative is a potent, selective, competitive, and orally active antagonist of vasopressin V2 receptor with an IC50 value of 14 nM. Mozavaptan hydrochloride shows ~85-fold selectivity for V2 receptor over V1 receptor. Mozavaptan hydrochloride has the potential for hyponatremia, syndrome of inappropriate antidiuretic hormone (SIADH), and congestive heart failure treatment.

Trivial name OPC 31260 HCl
Catalog Number E4957
Molecular Formula C16H14BrN5O4S.HCl
CAS# 138470-70-9
Inchi InChI=1S/C16H14BrN5O4S.ClH/c1-11-3-5-13(22(23)24)7-15(11)27(25,26)20(2)19-9-14-8-18-16-6-4-12(17)10-21(14)16;/h3-10H,1-2H3;1H/b19-9+;
Inchi Key VOUDEIAYNKZQKM-MYHMWQFYSA-N
SMILES CC1=C(C=C(C=C1)[N+](=O)[O-])S(=O)(=O)N(C)N=CC2=CN=C3N2C=C(C=C3)Br.Cl
Size 1g
Supplier Page http://www.selleckchem.com/products/mozavaptan-hydrochloride.html
Additional Information https://file.selleck.cn/downloads/struct/E4957-Mozavaptan-hydrochloride-chemical-structure.png